Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50045928
TargetUDP-glucuronosyltransferase 1A1(Human)
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  1.54E+3nMAssay Description:Substrate inhibition of human UGT1A1-mediated T-5224 acyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetUDP-glucuronosyltransferase 1A3(Human)
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  2.55E+3nMAssay Description:Substrate inhibition of human UGT1A3-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetUDP-glucuronosyltransferase 1A8(Human)
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  3.64E+3nMAssay Description:Substrate inhibition of human UGT1A8-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetUDP-glucuronosyltransferase 1A1(Human)
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  4.67E+3nMAssay Description:Substrate inhibition of human UGT1A1-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed
TargetUDP-glucuronosyltransferase 1A3(Human)
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  1.35E+4nMAssay Description:Substrate inhibition of human UGT1A3-mediated T-5224 acyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2016
Entry Details Article
PubMed