Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50033512
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346584(CHEMBL1795979)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346585(CHEMBL1795980 | S2101)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346586(CHEMBL1795981 | US8765820, 5a)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346589(CHEMBL255520 | CHEMBL1795974)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346583(CHEMBL1795978)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346591(CHEMBL1795982)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346582(CHEMBL1795977)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346590(CHEMBL1795975)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346594(CHEMBL1795976)
Affinity DataKi:  1.17E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human LSD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50113851(Tranylcypromine,(+) | TRANYLCYPROMINE | US8609708,...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataKi:  2.66E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataKi:  2.81E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346587(CHEMBL1795972)
Affinity DataKi:  4.18E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346588(CHEMBL1795973)
Affinity DataKi:  7.96E+4nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346592(CHEMBL1795983)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50346593(CHEMBL1795984)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged full length LSD1 expressed in Escherichia coli BL21 (DE3) assessed as inactivation constant preincubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataKi:  1.68E+5nMAssay Description:Inhibition of human truncated LSD1 lacking N-terminal 184 amino acidsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataKi:  1.68E+5nMAssay Description:Inhibition of human truncated LSD1 lacking N-terminal 184 amino acidsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed