Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50033371
TargetCystic fibrosis transmembrane conductance regulator(Human)
University Joseph Fourier-Grenoble 1/Cnrs

Curated by ChEMBL
LigandPNGBDBM50343996(2,4-dimethylpyrido[1,2-a]pyrimidin-5-ium-3-olate |...)
Affinity DataIC50: 5nMAssay Description:Inhibition of wild type CFTR expressed in CHO cells by [125I]iodide efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University Joseph Fourier-Grenoble 1/Cnrs

Curated by ChEMBL
LigandPNGBDBM50343998(CHEMBL1779954 | CHEMBL1779953 | (2S,3R,4R)-3,4-dih...)
Affinity DataIC50: 15nMAssay Description:Inhibition of wild type CFTR expressed in CHO cells by [125I]iodide efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University Joseph Fourier-Grenoble 1/Cnrs

Curated by ChEMBL
LigandPNGBDBM50343998(CHEMBL1779954 | CHEMBL1779953 | (2S,3R,4R)-3,4-dih...)
Affinity DataIC50: 15nMAssay Description:Inhibition of wild type CFTR expressed in CHO cells by [125I]iodide efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University Joseph Fourier-Grenoble 1/Cnrs

Curated by ChEMBL
LigandPNGBDBM50343997(2,4-dimethylpyrimido[2,1-a]isoquinolin-5-ium-3-ola...)
Affinity DataIC50: 16nMAssay Description:Inhibition of wild type CFTR expressed in CHO cells by [125I]iodide efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University Joseph Fourier-Grenoble 1/Cnrs

Curated by ChEMBL
LigandPNGBDBM50012957(1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfon...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of wild type CFTR expressed in CHO cells by [125I]iodide efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed