Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50033237
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM50341878((2R)-2-{[7-(benzylamino)-3-(propan-2-yl)-1H-pyrazo...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CDK2/cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM50341878((2R)-2-{[7-(benzylamino)-3-(propan-2-yl)-1H-pyrazo...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CDK7/cyclin H/MAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM50341878((2R)-2-{[7-(benzylamino)-3-(propan-2-yl)-1H-pyrazo...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant CDK5/p35More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant CDK2/cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human recombinant CDK7/cyclin H/MAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 940nMAssay Description:Inhibition of human recombinant CDK5/p35More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM50341878((2R)-2-{[7-(benzylamino)-3-(propan-2-yl)-1H-pyrazo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CDK9/cyclin T1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palacky£? University and Institute of Experimental Botany Ascr

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of human recombinant CDK9/cyclin T1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed