Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50004524
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50: 223nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50: 223nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50: 244nMAssay Description:Inhibition of HIV-1 reverse transcriptase K101E mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50175609(BDBM50192305 | 5-{3-[4-Amino-9-(tert-butyl-dimethy...)
Affinity DataIC50: 560nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50169035([2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D-ribo...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50483735(CHEMBL1766951)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: 1.65E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: 1.65E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase K101E mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus type 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50169035([2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D-ribo...)
Affinity DataIC50: 1.69E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed