Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50033384
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344231(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344230(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50333979(2-(3-(2-(2-(2,4-dichlorophenyl)-5-isopropyloxazol-...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344228(2-[3-[2-[2-(2,4-Dichlorophenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344231(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344227(2-[3-[2-[2-(4-Butylphenyl)-5-isopropyl-4-oxazolyl]...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344230(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344224(2-[3-[2-[2-(2-Hydroxyphenyl)-5-isopropyl-4-oxazoly...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344231(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  990nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344226(2-[3-[2-[2-(4-tert-Butylphenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344226(2-[3-[2-[2-(4-tert-Butylphenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344221(2-[3-[2-[2-(2-Chlorophenyl)-5-isopropyl-4-oxazolyl...)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344223(2-[3-[2-[2-(2-Chlorophenyl)-5-hexyl-4-oxazolyl]eth...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344223(2-[3-[2-[2-(2-Chlorophenyl)-5-hexyl-4-oxazolyl]eth...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344227(2-[3-[2-[2-(4-Butylphenyl)-5-isopropyl-4-oxazolyl]...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344226(2-[3-[2-[2-(4-tert-Butylphenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50:  2.90E+3nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344227(2-[3-[2-[2-(4-Butylphenyl)-5-isopropyl-4-oxazolyl]...)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344230(2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]...)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344220(2-[3-[2-[2-(2-Chlorophenyl)-5-propyl-4-oxazolyl]et...)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344223(2-[3-[2-[2-(2-Chlorophenyl)-5-hexyl-4-oxazolyl]eth...)
Affinity DataEC50:  5.90E+3nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344218(2-[3-[2-[5-Ethyl-2-phenyl-4-oxazolyl]ethyl]-1,2-be...)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344228(2-[3-[2-[2-(2,4-Dichlorophenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50:  8.60E+3nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344219(2-[3-[2-[2-Phenyl-5-propyl-4-oxazolyl]ethyl]-1,2-b...)
Affinity DataEC50:  9.80E+3nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344222(2-[3-[2-[5-tert-Butyl-2-(2-chlorophenyl)-4-oxazoly...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344222(2-[3-[2-[5-tert-Butyl-2-(2-chlorophenyl)-4-oxazoly...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50333979(2-(3-(2-(2-(2,4-dichlorophenyl)-5-isopropyloxazol-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50333979(2-(3-(2-(2-(2,4-dichlorophenyl)-5-isopropyloxazol-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344222(2-[3-[2-[5-tert-Butyl-2-(2-chlorophenyl)-4-oxazoly...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344225(2-[3-[2-[5-Isopropyl-2-[2-(trifluoromethyl)phenyl]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344225(2-[3-[2-[5-Isopropyl-2-[2-(trifluoromethyl)phenyl]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344225(2-[3-[2-[5-Isopropyl-2-[2-(trifluoromethyl)phenyl]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344229(2-[3-[2-[2-(2,6-Dichlorophenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344229(2-[3-[2-[2-(2,6-Dichlorophenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344229(2-[3-[2-[2-(2,6-Dichlorophenyl)-5-isopropyl-4-oxaz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344224(2-[3-[2-[2-(2-Hydroxyphenyl)-5-isopropyl-4-oxazoly...)
Affinity DataEC50:  1.04E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344217(2-[3-[2-[5-Methyl-2-phenyl-4-oxazolyl]ethyl]-1,2-b...)
Affinity DataEC50:  1.29E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344219(2-[3-[2-[2-Phenyl-5-propyl-4-oxazolyl]ethyl]-1,2-b...)
Affinity DataEC50:  1.32E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50344220(2-[3-[2-[2-(2-Chlorophenyl)-5-propyl-4-oxazolyl]et...)
Affinity DataEC50:  1.39E+4nMAssay Description:Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
Displayed 1 to 50 (of 60 total ) | Next | Last >>
Jump to: