Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 50001148
LigandPNGBDBM50013184(CHEMBL343066 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013209(CHEMBL140365 | 4-Chloro-N-[5-(2-fluoro-phenyl)-1-m...)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50452659(CHEMBL304546)
Affinity DataIC50: 1.10nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013185(CHEMBL141354 | 2-Benzo[b]thiophen-4-yl-N-[5-(2-flu...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013208(CHEMBL337530 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 8nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50013182(CHEMBL141365 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 8.60nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013191(CHEMBL141629 | 3-{[5-(2-Fluoro-phenyl)-1-methyl-2,...)
Affinity DataIC50: 18nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013191(CHEMBL141629 | 3-{[5-(2-Fluoro-phenyl)-1-methyl-2,...)
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013199(CHEMBL342415 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50452659(CHEMBL304546)
Affinity DataIC50: 29nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013195(CHEMBL140749 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013188(CHEMBL141786 | 2-Amino-N-[5-(2-fluoro-phenyl)-1-me...)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049805(Tifluadom | Thiophene-3-carboxylic acid [5-(2-fluo...)
Affinity DataIC50: 47nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50452658(CHEMBL68870)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013192(CHEMBL140495 | [5-(2-Fluoro-phenyl)-2,3-dihydro-1H...)
Affinity DataIC50: 91nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013204(CHEMBL343158 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 93nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013205(CHEMBL141048 | 2-(Acetylamino-methylsulfanyl)-N-[5...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013184(CHEMBL343066 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 160nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 245nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type B receptor in guinea pig brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50452658(CHEMBL68870)
Affinity DataIC50: 260nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013197(CHEMBL140620 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 450nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013185(CHEMBL141354 | 2-Benzo[b]thiophen-4-yl-N-[5-(2-flu...)
Affinity DataIC50: 450nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013203(CHEMBL344154 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 540nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013208(CHEMBL337530 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 600nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013209(CHEMBL140365 | 4-Chloro-N-[5-(2-fluoro-phenyl)-1-m...)
Affinity DataIC50: 800nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013199(CHEMBL342415 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013200(CHEMBL141051 | [5-(2-Fluoro-phenyl)-1-methyl-2,3-d...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013187(CHEMBL139615 | 2-Fluoro-N-[5-(2-fluoro-phenyl)-1-m...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013182(CHEMBL141365 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013190(CHEMBL342256 | [1-{[5-(2-Fluoro-phenyl)-1-methyl-2...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013207(CHEMBL140516 | 2-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013195(CHEMBL140749 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013179(CHEMBL336690 | [5-(2-Fluoro-phenyl)-1-methyl-2,3-d...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013203(CHEMBL344154 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013183(CHEMBL140984 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 7.50E+3nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013186(CHEMBL140974 | (Diastereomer)-N-[5-(2-Fluoro-pheny...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluated for its concentration required for displacement of [3H]-Naloxone from opioid receptors in rat brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013197(CHEMBL140620 | N-[5-(2-Fluoro-phenyl)-1-methyl-2,3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013204(CHEMBL343158 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013188(CHEMBL141786 | 2-Amino-N-[5-(2-fluoro-phenyl)-1-me...)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013189(CHEMBL334933 | [5-(2-Fluoro-phenyl)-2-oxo-2,3-dihy...)
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [3H]dihydromorphine (DHM) from rat brain Opioid receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013194(CHEMBL139520 | 3,3,3-Trifluoro-N-[5-(2-fluoro-phen...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013196(CHEMBL341815 | Bis[5-(2-fluoro-phenyl)-1,3-dihydro...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013202(CHEMBL423918 | 3-[(5-Chloro-pyrazin-2-ylamino)-met...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013184(CHEMBL343066 | 1H-Indole-2-carboxylic acid [5-(2-f...)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type B receptor in guinea pig brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013183(CHEMBL140984 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013189(CHEMBL334933 | [5-(2-Fluoro-phenyl)-2-oxo-2,3-dihy...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013185(CHEMBL141354 | 2-Benzo[b]thiophen-4-yl-N-[5-(2-flu...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type B receptor in guinea pig brain tissuesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50013181(CHEMBL336256 | (2-(Acetylamino-methylsulfanyl)-1-{...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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