Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50033448
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50345548([13C,15N-Y,P,V]cyclic CRYPEVEIC | cyclic CRYPEVEIC...)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of human GST-tagged-Pin1 PPIase activity using WFYpSPR-pNA as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50345548([13C,15N-Y,P,V]cyclic CRYPEVEIC | cyclic CRYPEVEIC...)
Affinity DataKi:  520nMAssay Description:Inhibition of human GST-tagged-Pin1 PPIase activity using Suc-AEPF-pNA as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50345549(CRYPEVEIC | CHEMBL1784539)
Affinity DataKi:  4.40E+4nMAssay Description:Inhibition of human GST-tagged-Pin1 PPIase activity using Suc-AEPF-pNA as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed