Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50033422
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM20880(CHEMBL429910 | C-aryl glucoside, 6 | BMS-512148 | ...)
Affinity DataIC50: 1.35nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345019((2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(4-(pent-2...)
Affinity DataIC50: 59.5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345022((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(15-oxa-tricycl...)
Affinity DataIC50: 81.9nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345020((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(15-oxa-tricycl...)
Affinity DataIC50: 89.6nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345023((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(16-oxa-tricycl...)
Affinity DataIC50: 99.7nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetSolute carrier family 5 member 4(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345021((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(16-oxa-tricycl...)
Affinity DataIC50: 103nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed