Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50033760
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50350791(LEVOBUPIVACAINE HYDROCHLORIDE)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50350791(LEVOBUPIVACAINE HYDROCHLORIDE)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in CHO cells by whole-cell patch clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50350790(Bupivacaine | BUPIVACAINE HYDROCHLORIDE | SAMPL3, ...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in CHO cells by whole-cell patch clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50350790(Bupivacaine | BUPIVACAINE HYDROCHLORIDE | SAMPL3, ...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50350789(CHEMBL189827 | BUPIVACAINE)
Affinity DataIC50: 8.40E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed