Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50033549
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347195(CHEMBL1795747)
Affinity DataIC50: 96nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347200(CHEMBL1795752)
Affinity DataIC50: 190nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50098126(LY-293646 | 2-morpholino-4H-benzo[h]chromen-4-one ...)
Affinity DataIC50: 300nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347198(CHEMBL1795750)
Affinity DataIC50: 330nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50159668(2-Morpholin-4-yl-benzo[g]chromen-4-one | 2-morphol...)
Affinity DataIC50: 400nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347191(CHEMBL1795743)
Affinity DataIC50: 420nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347194(CHEMBL1795746)
Affinity DataIC50: 717nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347190(CHEMBL1795742)
Affinity DataIC50: 720nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347199(CHEMBL1795751)
Affinity DataIC50: 760nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347197(CHEMBL1795749)
Affinity DataIC50: 930nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347196(CHEMBL1795748)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347193(CHEMBL1795745)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347201(CHEMBL1795753)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347192(CHEMBL1795744)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed