Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50034164
TargetHistone deacetylase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant full-length HDAC1 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human recombinant full-length HDAC1 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50: 12.7nMAssay Description:Inhibition of human recombinant full-length HDAC2 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant full-length HDAC2 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 21.8nMAssay Description:Inhibition of human recombinant full-length HDAC3 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50: 23.9nMAssay Description:Inhibition of human recombinant full-length HDAC3 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50: 50.2nMAssay Description:Inhibition of human recombinant full-length HDAC6 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 57.3nMAssay Description:Inhibition of human recombinant full-length HDAC6 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed