Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 50041933
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  794nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50318159(CHEMBL1095777 | 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50318159(CHEMBL1095777 | 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418939(CHEMBL1807873)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418955(CHEMBL1807831)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418947(CHEMBL1807874)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418950(CHEMBL1807832)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418958(CHEMBL1807820)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418946(CHEMBL1807817)
Affinity DataEC50:  0.0631nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418944(CHEMBL1807819)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM86453(NSC_3083544 | CAS_73573-87-2 | Formoterol)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418945(CHEMBL1807818)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418938(CHEMBL1807872)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418944(CHEMBL1807819)
Affinity DataEC50:  4nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418954(CHEMBL1807827)
Affinity DataEC50:  100nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418953(CHEMBL1807828)
Affinity DataEC50:  100nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418952(CHEMBL1807829)
Affinity DataEC50:  100nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418951(CHEMBL1807830)
Affinity DataEC50:  40nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418950(CHEMBL1807832)
Affinity DataEC50:  32nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418947(CHEMBL1807874)
Affinity DataEC50:  200nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418939(CHEMBL1807873)
Affinity DataEC50:  158nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418938(CHEMBL1807872)
Affinity DataEC50:  40nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418948(CHEMBL1807870)
Affinity DataEC50:  40nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418949(CHEMBL1807869)
Affinity DataEC50:  100nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418951(CHEMBL1807830)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418956(CHEMBL1807826)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418949(CHEMBL1807869)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418940(CHEMBL1807825)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418948(CHEMBL1807870)
Affinity DataEC50:  0.398nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418941(CHEMBL1807823)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418937(CHEMBL1807871)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418942(CHEMBL1807822)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418943(CHEMBL1807821)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418953(CHEMBL1807828)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418954(CHEMBL1807827)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418952(CHEMBL1807829)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418957(CHEMBL1807824)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50128690(SB-07499 | 4-Hydroxy-7-{2-[2-(3-phenethyloxy-propa...)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418937(CHEMBL1807871)
Affinity DataEC50:  63nMAssay Description:Agonist activity at adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418943(CHEMBL1807821)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418942(CHEMBL1807822)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418944(CHEMBL1807819)
Affinity DataIC50: 4nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418958(CHEMBL1807820)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418945(CHEMBL1807818)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418946(CHEMBL1807817)
Affinity DataIC50: 7.90nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418948(CHEMBL1807870)
Affinity DataIC50: 40nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418957(CHEMBL1807824)
Affinity DataIC50: 50nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418939(CHEMBL1807873)
Affinity DataIC50: 50nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50418938(CHEMBL1807872)
Affinity DataIC50: 63nMAssay Description:Binding affinity to adrenergic beta1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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