Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50034305
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataIC50: 9.5nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataIC50: 15.7nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  59.8nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360274(CHEMBL1933101)
Affinity DataIC50: 107nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  169nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50: 197nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataIC50: 313nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360272(CHEMBL1933099)
Affinity DataIC50: 317nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360277(CHEMBL1933108)
Affinity DataIC50: 419nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360278(CHEMBL1933109)
Affinity DataIC50: 717nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  973nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  1.53E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed