Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50033659
TargetTranscription factor Jun(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50349193(CHEMBL1807644)
Affinity DataEC50:  1.49E+3nMAssay Description:Inhibition of TPA-induced AP-1 activity expressed in human HEK293T cells treated 1 hr before TPA challenge measured after 18 hrs by FRET based beta-l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50349194(NSC-14975 | GLAUCARUBINONE)
Affinity DataEC50:  130nMAssay Description:Inhibition of TPA-induced AP-1 activity expressed in human HEK293T cells treated 1 hr before TPA challenge measured after 18 hrs by FRET based beta-l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed