Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50004563
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50: 5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50087419(2-(3,4-dihydroxy-5-methoxystyryl)-8-hydroxyquinoli...)
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50087419(2-(3,4-dihydroxy-5-methoxystyryl)-8-hydroxyquinoli...)
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484136(CHEMBL1813126)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484142(CHEMBL1813127)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484137(CCDC 752665 | CHEMBL1682442)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484141(CHEMBL1456957)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484138(CHEMBL1813133)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50065794(8-Hydroxy-2-methyl-quinoline-7-carboxylic acid | 8...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484134(CHEMBL1813129)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484135(CHEMBL1813128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484139(CHEMBL1813131)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Silesia

Curated by ChEMBL
LigandPNGBDBM50484140(CHEMBL1813134)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of HIV1 recombinant integrase 3'-processing and strand transfer activity using 21-mer U5B/U5A duplex oligonucleotides after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed