Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50039472
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350712(CHEMBL1812084)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350706(CHEMBL1811922)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein TraR(Agrobacterium tumefaciens)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350704(CHEMBL1814829)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350709(CHEMBL1812080)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350708(CHEMBL1814832)
Affinity DataIC50: 310nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350711(CHEMBL1812089)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350704(CHEMBL1814829)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350710(CHEMBL1812087)
Affinity DataIC50: 770nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350707(CHEMBL1814831)
Affinity DataIC50: 840nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein TraR(Agrobacterium tumefaciens)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein TraR(Agrobacterium tumefaciens)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350706(CHEMBL1811922)
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein TraR(Agrobacterium tumefaciens)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein TraR(Agrobacterium tumefaciens)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350708(CHEMBL1814832)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2013
Entry Details Article
PubMed