Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50033787
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351253(CHEMBL1818528)
Affinity DataEC50:  160nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351254(CHEMBL1818529)
Affinity DataEC50:  115nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM23772(STLC | Tritylcysteine | 3-Tritylthio-L-alanine | N...)
Affinity DataEC50:  1.72E+3nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM23823((2R)-2-amino-3-{[(4-methoxyphenyl)diphenylmethyl]s...)
Affinity DataEC50:  230nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351255(CHEMBL1818525)
Affinity DataEC50:  600nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351256(CHEMBL1818526)
Affinity DataEC50:  294nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351257(CHEMBL1818527)
Affinity DataEC50:  190nMAssay Description:Inhibition of KSP in human HeLa cells assessed as bipolar spindle formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351257(CHEMBL1818527)
Affinity DataIC50: 127nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351253(CHEMBL1818528)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351254(CHEMBL1818529)
Affinity DataIC50: 136nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351255(CHEMBL1818525)
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM23823((2R)-2-amino-3-{[(4-methoxyphenyl)diphenylmethyl]s...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM50351256(CHEMBL1818526)
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
New Mexico State University

Curated by ChEMBL
LigandPNGBDBM23772(STLC | Tritylcysteine | 3-Tritylthio-L-alanine | N...)
Affinity DataIC50: 620nMAssay Description:Inhibition of human recombinant microtubule-activated KSP motor domain ATPase activity after 10 mins by end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed