Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 5655
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM92463(Imipenem)
Affinity DataKi:  3.20E+3nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM50140672(Beta-lactam compound, 2 | CHEMBL25613 | (2S,5R,6R)...)
Affinity DataKi:  3.00E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM92461(Beta-lactam compound, 4)
Affinity DataKi:  4.20E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM92464(Carbenicillin)
Affinity DataKi:  7.80E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM50140671(CHEMBL277857 | Beta-lactam compound, 1 | (2S,5R,6S...)
Affinity DataKi:  8.30E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
York University

LigandPNGBDBM92462(Beta-lactam compound, 3)
Affinity DataKi:  4.04E+5nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed