Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50033984
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354986(CHEMBL1834889)
Affinity DataEC50:  19.4nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354987(CHEMBL1834890)
Affinity DataEC50:  1.11nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354988(CHEMBL1834891)
Affinity DataEC50:  0.920nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354989(CHEMBL1834892)
Affinity DataEC50:  1.25nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354990(CHEMBL1834893)
Affinity DataEC50:  0.0600nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50354991(CHEMBL1834894)
Affinity DataEC50:  1.29nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50329706((2S)-3-{4-[1-ethyl-1-(4-{[(2R)-2-hydroxy-3,3-dimet...)
Affinity DataEC50:  0.0400nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0100nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed