Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50034108
LigandPNGBDBM50067133(CHEMBL631 | 1-[2-(2-Hydroxy-3-propylamino-propoxy)...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human kir6.2/SUR2A ion channel coexpressed in human HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357206(CHEMBL1915083 | CHEMBL1962378)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human cloned ERG channel expressed in chinese hamster CHO cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50067133(CHEMBL631 | 1-[2-(2-Hydroxy-3-propylamino-propoxy)...)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of human cloned ERG channel expressed in chinese hamster CHO cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50067133(CHEMBL631 | 1-[2-(2-Hydroxy-3-propylamino-propoxy)...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as tonic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357204(CHEMBL1914835 | CHEMBL1963280)
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of human cloned ERG channel expressed in chinese hamster CHO cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357205(CHEMBL1963594 | CHEMBL1914844)
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of human cloned ERG channel expressed in chinese hamster CHO cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357207(CHEMBL1915364 | CHEMBL1963307)
Affinity DataIC50: 4.84E+3nMAssay Description:Inhibition of human cloned ERG channel expressed in chinese hamster CHO cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50357207(CHEMBL1915364 | CHEMBL1963307)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human kir6.2/SUR2A ion channel coexpressed in human HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50357205(CHEMBL1963594 | CHEMBL1914844)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human kir6.2/SUR2A ion channel coexpressed in human HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50357204(CHEMBL1914835 | CHEMBL1963280)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human kir6.2/SUR2A ion channel coexpressed in human HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357207(CHEMBL1915364 | CHEMBL1963307)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as phasic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357205(CHEMBL1963594 | CHEMBL1914844)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as phasic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357204(CHEMBL1914835 | CHEMBL1963280)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as phasic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50067133(CHEMBL631 | 1-[2-(2-Hydroxy-3-propylamino-propoxy)...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as phasic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357207(CHEMBL1915364 | CHEMBL1963307)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as tonic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357205(CHEMBL1963594 | CHEMBL1914844)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as tonic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50357204(CHEMBL1914835 | CHEMBL1963280)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human cloned Nav1.5 channel expressed in chinese hamster CHO cells assessed as tonic inhibition after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed