Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50004591
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484478(CHEMBL1929019 | jm5b01461, Compound 47)
Affinity DataIC50: 65nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484484(CHEMBL1929023)
Affinity DataIC50: 98nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484483(CHEMBL1929020 | acs.jmedchem.1c00409_ST.132)
Affinity DataIC50: 270nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484491(CHEMBL1929022 | acs.jmedchem.1c00409_ST.144)
Affinity DataIC50: 340nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484487(CHEMBL1929018 | acs.jmedchem.1c00409_ST.150)
Affinity DataIC50: 390nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484482(CHEMBL1929017 | med.21724, Compound 45 | acs.jmedc...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484482(CHEMBL1929017 | med.21724, Compound 45 | acs.jmedc...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484490(CHEMBL1929021 | acs.jmedchem.1c00409_ST.508)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 measured after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484479(CHEMBL479724 | med.21724, Compound 44 | acs.jmedch...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484485(CHEMBL1929016 | acs.jmedchem.1c00409_ST.700)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484488(CHEMBL1929015 | acs.jmedchem.1c00409_ST.720)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484489(CHEMBL1929009)
Affinity DataIC50: 3.30E+5nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484480(CHEMBL1929012)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484481(CHEMBL1929014 | acs.jmedchem.1c00409_ST.815)
Affinity DataIC50: 2.00E+6nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetChymotrypsin-like protease CTRL-1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50484486(CHEMBL1929013)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of chymotrypsin-like protease R188I mutant using peptide substrate SO1 preincubated for 20 mins before substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed