Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 5485
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86654(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 1)
Affinity DataIC50: 67nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86648(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5b)
Affinity DataIC50: 6.40E+3nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86653(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5g)
Affinity DataIC50: 6.50E+3nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86647(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5a)
Affinity DataIC50: 6.70E+3nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86651(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5e)
Affinity DataIC50: 7.10E+3nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86652(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5f)
Affinity DataIC50: 1.23E+4nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86650(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5d)
Affinity DataIC50: 1.56E+4nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [1148-1435](Human immunodeficiency virus type 1)
National Institutes of Health

LigandPNGBDBM86649(Bicyclic hydroxy-1H-pyrrolopyridine-trione, 5c)
Affinity DataIC50: 2.16E+4nMAssay Description:The compound were evaluated in biochemical IN (integrase) assay that measure inhibitory potency (IC50 values)against both the 3'-processing(3'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2012
Entry Details Article
PubMed