Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50039872
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKd: 350nMAssay Description:Binding affinity to PA N-terminal domain (Direct)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 860nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 960nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 990nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.39E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.65E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.84E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.97E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 2.07E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.28E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.44E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.22E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.50E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.50E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 3.56E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.56E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.66E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.70E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.80E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 4.85E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 5.41E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 5.52E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 5.92E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 6.70E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 6.80E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 6.80E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 7.67E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 8.17E+3nMAssay Description:Plaque growth inhibitionMore data for this Ligand-Target Pair
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.12E+4nMAssay Description:Binding affinity to PA N-terminal domain (Competitive)More data for this Ligand-Target Pair







3D Structure (crystal)



















