Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50034564
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364312(CHEMBL1949764)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364311(CHEMBL1949763)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364323(CHEMBL1949928)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364323(CHEMBL1949928)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364309(CHEMBL1949761)
Affinity DataIC50: 133nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364310(CHEMBL1949762)
Affinity DataIC50: 135nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364308(CHEMBL1949760)
Affinity DataIC50: 179nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364313(CHEMBL1949765)
Affinity DataIC50: 227nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364320(CHEMBL1949772)
Affinity DataIC50: 245nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364315(CHEMBL1949767)
Affinity DataIC50: 281nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364316(CHEMBL1949768)
Affinity DataIC50: 306nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364314(CHEMBL1949766)
Affinity DataIC50: 357nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364322(CHEMBL1949927)
Affinity DataIC50: 790nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364322(CHEMBL1949927)
Affinity DataIC50: 790nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364321(CHEMBL1949773)
Affinity DataIC50: 1.36E+3nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364321(CHEMBL1949773)
Affinity DataIC50: 1.36E+3nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in human astrocytoma cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of M1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of NA transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of M4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of CYP 3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of DA transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of CYP 2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP 2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP 1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP 2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50361052(CHEMBL1949758 | CHEMBL1935589)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364323(CHEMBL1949928)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364323(CHEMBL1949928)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364312(CHEMBL1949764)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364311(CHEMBL1949763)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364310(CHEMBL1949762)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364316(CHEMBL1949768)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364311(CHEMBL1949763)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364311(CHEMBL1949763)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364316(CHEMBL1949768)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364316(CHEMBL1949768)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364326(CHEMBL1949930)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364308(CHEMBL1949760)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364313(CHEMBL1949765)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364309(CHEMBL1949761)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364312(CHEMBL1949764)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364314(CHEMBL1949766)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50364324(CHEMBL1949677)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
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