Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50034459
TargetVasopressin V1a receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362873(CHEMBL1940587)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362871(CHEMBL1940588)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362872(CHEMBL1940586)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]arginine-vasopressin from human Vasopressin V1a receptor after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362872(CHEMBL1940586)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362872(CHEMBL1940586)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human V1b receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362873(CHEMBL1940587)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity to human V1b receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362871(CHEMBL1940588)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human V1b receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362873(CHEMBL1940587)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Lehigh University

Curated by ChEMBL
LigandPNGBDBM50362871(CHEMBL1940588)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed