Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50040141
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389772(CHEMBL2070244)
Affinity DataEC50:  0.470nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389780(CHEMBL2069317)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389781(CHEMBL2070254)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389782(CHEMBL2070374)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389769(BREMELANOTIDE)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389770(CHEMBL2070242)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389776(CHEMBL2070249)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389773(CHEMBL2070246)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389774(CHEMBL2070247)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389775(CHEMBL2070248)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389777(CHEMBL2070250)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389778(CHEMBL2070251)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389779(CHEMBL2070252)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389778(CHEMBL2070251)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389773(CHEMBL2070246)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389780(CHEMBL2069317)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389776(CHEMBL2070249)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389777(CHEMBL2070250)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389774(CHEMBL2070247)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389769(BREMELANOTIDE)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389779(CHEMBL2070252)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389775(CHEMBL2070248)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  0.370nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  0.470nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.480nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389782(CHEMBL2070374)
Affinity DataKi:  0.580nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.780nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389772(CHEMBL2070244)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389773(CHEMBL2070246)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389780(CHEMBL2069317)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389778(CHEMBL2070251)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389775(CHEMBL2070248)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389779(CHEMBL2070252)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389772(CHEMBL2070244)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389770(CHEMBL2070242)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389770(CHEMBL2070242)
Affinity DataKi:  5.10nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389769(BREMELANOTIDE)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389785(CHEMBL2070373)
Affinity DataKi:  7.80nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
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