Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50034654
TargetSodium-dependent dopamine transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat DAT-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat DAT-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat NET-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat NET-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of CYP3A4 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of CYP3A5 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of CYP3A4 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of CYP3A5 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of CYP2C19 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of CYP2C19 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.77E+5nMAssay Description:Inhibition of CYP2D6 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 1.77E+5nMAssay Description:Inhibition of CYP2D6 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 2.33E+5nMAssay Description:Inhibition of CYP2C9 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 2.33E+5nMAssay Description:Inhibition of CYP2C9 in human microsomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat SERT-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of rat SERT-mediated uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed