Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50039610
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50326618([11C]-3-(2-methoxyethyl)-4,5-dimethyl-3H-thiazol-(...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380894(CHEMBL2019078)
Affinity DataIC50: 1nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380894(CHEMBL2019078)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380896(CHEMBL2019081)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380896(CHEMBL2019081)
Affinity DataIC50: 7nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380887(CHEMBL2019083)
Affinity DataIC50: 7nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380889(CHEMBL2019086)
Affinity DataIC50: 9nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380900(CHEMBL2019080)
Affinity DataIC50: 14nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380889(CHEMBL2019086)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataIC50: 24nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataIC50: 51nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380900(CHEMBL2019080)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380887(CHEMBL2019083)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380896(CHEMBL2019081)
Affinity DataIC50: 76nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380900(CHEMBL2019080)
Affinity DataIC50: 113nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380890(CHEMBL2019087)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380895(CHEMBL2019079)
Affinity DataKi:  177nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380896(CHEMBL2019081)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380897(CHEMBL2019084)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380900(CHEMBL2019080)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380893(CHEMBL2019091)
Affinity DataKi:  263nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380889(CHEMBL2019086)
Affinity DataKi:  266nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380888(CHEMBL2019092)
Affinity DataKi:  294nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380899(CHEMBL2019088)
Affinity DataKi:  348nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380852(CHEMBL2018656)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380891(CHEMBL2019089)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380894(CHEMBL2019078)
Affinity DataIC50: 468nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380889(CHEMBL2019086)
Affinity DataIC50: 514nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380894(CHEMBL2019078)
Affinity DataKi:  793nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380895(CHEMBL2019079)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380852(CHEMBL2018656)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380887(CHEMBL2019083)
Affinity DataIC50: 2.00E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataIC50: 2.00E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataIC50: 2.00E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380898(CHEMBL2019085)
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataKi:  3.06E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380890(CHEMBL2019087)
Affinity DataKi:  3.95E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380892(S-777469 | CHEMBL2019090)
Affinity DataKi:  4.07E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380888(CHEMBL2019092)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380887(CHEMBL2019083)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380897(CHEMBL2019084)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380891(CHEMBL2019089)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380893(CHEMBL2019091)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed