Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50034689
TargetNuclear receptor subfamily 1 group D member 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50: 560nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50: 620nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50: 670nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50: 710nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50: 790nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataKd:  800nMAssay Description:Dissociation constant for binding to REV-ERB-alpha by circular dichroismMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50: 800nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed