Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50040853
TargetHistamine H3 receptor(Rat)
Eth Zurich (Swiss Federal Institute of Technology)

Curated by ChEMBL
LigandPNGBDBM50278350(CHEMBL513193 | CHEMBL2203701 | 4-fluoro-1-(4-(3-(p...)
Affinity DataKd:  0.340nMAssay Description:Binding affinity to rat brain histamine H3 receptor after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Eth Zurich (Swiss Federal Institute of Technology)

Curated by ChEMBL
LigandPNGBDBM50278350(CHEMBL513193 | CHEMBL2203701 | 4-fluoro-1-(4-(3-(p...)
Affinity DataKd: >3.00E+3nMAssay Description:Binding affinity to rat histamine H3 receptor low affinity site after 1 hr by Schard plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Eth Zurich (Swiss Federal Institute of Technology)

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  0.575nMAssay Description:Binding affinity to human recombinant histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Eth Zurich (Swiss Federal Institute of Technology)

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataKi:  0.654nMAssay Description:Binding affinity to rat cerebral cortex histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Eth Zurich (Swiss Federal Institute of Technology)

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  1.26nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed