Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50039670
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382082(CHEMBL2022130)
Affinity DataEC50:  290nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382073(CHEMBL2024616)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382074(CHEMBL2024617)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382075(CHEMBL2024618)
Affinity DataEC50:  26nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382076(CHEMBL2024619)
Affinity DataEC50:  6.20nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382077(CHEMBL2022125)
Affinity DataEC50:  7.40nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382078(CHEMBL2022126)
Affinity DataEC50:  80nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382079(CHEMBL2022127)
Affinity DataEC50:  59nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382080(CHEMBL2022128)
Affinity DataEC50:  320nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382081(CHEMBL2022129)
Affinity DataEC50:  15nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382072(CHEMBL2024615)
Affinity DataEC50:  190nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382083(CHEMBL2022131)
Affinity DataEC50:  32nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382084(CHEMBL2022132)
Affinity DataEC50:  38nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382085(CHEMBL2022133)
Affinity DataEC50:  48nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382086(CHEMBL2022134)
Affinity DataEC50:  4.5nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382087(CHEMBL2021930)
Affinity DataEC50:  1.10nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382055(CHEMBL2024606)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARalpha expressed in african green monkey COS1 cells after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382088(CHEMBL2024613)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382055(CHEMBL2024606)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARdelta expressed in african green monkey COS1 cells after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382055(CHEMBL2024606)
Affinity DataEC50:  15nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382056(CHEMBL2022743)
Affinity DataEC50:  61nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382057(CHEMBL2022744)
Affinity DataEC50:  2.60nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382058(CHEMBL2022745)
Affinity DataEC50:  1.5nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382059(CHEMBL2022746)
Affinity DataEC50:  6.90nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382060(CHEMBL2022747)
Affinity DataEC50:  3.40nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382061(CHEMBL2022748)
Affinity DataEC50:  11nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382062(CHEMBL2024604)
Affinity DataEC50:  32nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382063(CHEMBL2024605)
Affinity DataEC50:  8.60nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382064(CHEMBL2024607)
Affinity DataEC50:  2.30nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382065(CHEMBL2024608)
Affinity DataEC50:  3.10nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382066(CHEMBL2024609)
Affinity DataEC50:  5.5nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382067(CHEMBL2021928)
Affinity DataEC50:  5.20nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382068(CHEMBL2024610)
Affinity DataEC50:  6.70nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382069(CHEMBL2024611)
Affinity DataEC50:  10nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382070(CHEMBL2024612)
Affinity DataEC50:  94nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382071(CHEMBL2024614)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of human PPARgamma1 expressed in CHO-K1 cells co-expressing RXRalpha and PPRE after 1 day by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50382055(CHEMBL2024606)
Affinity DataIC50: 330nMAssay Description:Displacement of [3H]-AD-5061 from human GST-tagged PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed