Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50039842
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50384998(XANTHOHUMOL | CVD-0019905)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human PDK1 assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50252521(isoxanthohumol | CHEMBL492828)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of human PKC theta assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50252521(isoxanthohumol | CHEMBL492828)
Affinity DataIC50: 4.53E+4nMAssay Description:Inhibition of human PKC alpha assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50252521(isoxanthohumol | CHEMBL492828)
Affinity DataIC50: 5.87E+4nMAssay Description:Inhibition of human PDK1 assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50384998(XANTHOHUMOL | CVD-0019905)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PKC alpha assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50384998(XANTHOHUMOL | CVD-0019905)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PKC theta assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed