Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50039958
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P3 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  55nMAssay Description:Agonist activity against human S1P1 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  55nMAssay Description:Agonist activity against human S1P1 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  123nMAssay Description:Agonist activity against human S1P1 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  123nMAssay Description:Agonist activity against human S1P1 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P2 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P2 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P2 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P3 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P3 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P3 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386854(CHEMBL2048288)
Affinity DataEC50:  157nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  239nMAssay Description:Agonist activity against human S1P4 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  239nMAssay Description:Agonist activity against human S1P4 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P4 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P4 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  11nMAssay Description:Agonist activity against human S1P5 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  11nMAssay Description:Agonist activity against human S1P5 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  289nMAssay Description:Agonist activity against human S1P5 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  289nMAssay Description:Agonist activity against human S1P5 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386864(CHEMBL2048298)
Affinity DataEC50:  0.610nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity against human S1P2 by beta arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity against mouse S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386855(CHEMBL2048289)
Affinity DataEC50:  76nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386856(CHEMBL2048290)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386857(CHEMBL2048291)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386858(CHEMBL2048292)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386860(CHEMBL2048294)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386861(CHEMBL2048295)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386862(CHEMBL2048296)
Affinity DataEC50:  0.590nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386863(CHEMBL2048297)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  1.73nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity against mouse S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity against mouse S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Mouse)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity against mouse S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity against rat S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity against rat S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity against rat S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity against rat S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  0.760nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386853(CHEMBL2048287)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity against human S1P1 assessed as accumulation of cAMP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50386859(CHEMBL2048293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by astemizole assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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