Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50040405
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393724(CHEMBL2159120)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182946(4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazo...)
Affinity DataEC50:  135nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393724(CHEMBL2159120)
Affinity DataEC50:  61nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182939((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataEC50:  2nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataEC50:  27nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182946(4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazo...)
Affinity DataEC50:  9nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182943(4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazo...)
Affinity DataEC50:  161nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50154036(2-Amino-3-(4-hydroxy-phenyl)-1-[3-(4-phenyl-1H-imi...)
Affinity DataEC50:  2.45E+3nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50154036(2-Amino-3-(4-hydroxy-phenyl)-1-[3-(4-phenyl-1H-imi...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182943(4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazo...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182939((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393722(CHEMBL2159119)
Affinity DataEC50:  35nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393719(CHEMBL2159118)
Affinity DataEC50:  20nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393725(CHEMBL2159117)
Affinity DataEC50:  103nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataEC50:  1nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at kappa opioid receptor guinea pig colon tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393725(CHEMBL2159117)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393719(CHEMBL2159118)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182939((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182943(4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazo...)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393717(CHEMBL2159116)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393716(CHEMBL2159115)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182946(4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazo...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393721(CHEMBL2159114)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393722(CHEMBL2159119)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393724(CHEMBL2159120)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50154036(2-Amino-3-(4-hydroxy-phenyl)-1-[3-(4-phenyl-1H-imi...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393724(CHEMBL2159120)
Affinity DataKi:  1nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393725(CHEMBL2159117)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182943(4-((S)-2-amino-3-oxo-3-((S)-3-(4-phenyl-1H-imidazo...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393719(CHEMBL2159118)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182939((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393722(CHEMBL2159119)
Affinity DataKi:  12nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393727(CHEMBL2159113)
Affinity DataKi:  13nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50182946(4-((S)-2-amino-3-oxo-3-((S)-2-(4-phenyl-1H-imidazo...)
Affinity DataKi:  14nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393717(CHEMBL2159116)
Affinity DataKi:  15nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393716(CHEMBL2159115)
Affinity DataKi:  15nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393718(CHEMBL2159111)
Affinity DataKi:  17nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393721(CHEMBL2159114)
Affinity DataKi:  26nMAssay Description:Binding affinity to rat delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50154036(2-Amino-3-(4-hydroxy-phenyl)-1-[3-(4-phenyl-1H-imi...)
Affinity DataKi:  55nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50393720(CHEMBL2159122 | CHEMBL3216329)
Affinity DataKi:  55nMAssay Description:Binding affinity to guinea pig kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: