Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50040009
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387812(CHEMBL2058372)
Affinity DataIC50: 8.5nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387812(CHEMBL2058372)
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50061101(4-tert-butyl-N-[6-(2-hydroxyethoxy)-5-(2-methoxyph...)
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387811(CHEMBL2058371)
Affinity DataIC50: 9.10nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387811(CHEMBL2058371)
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387805(CHEMBL2058373)
Affinity DataIC50: 9.60nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387810(CHEMBL2058370)
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387813(CHEMBL2058374)
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387805(CHEMBL2058373)
Affinity DataIC50: 9.80nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387810(CHEMBL2058370)
Affinity DataIC50: 9.90nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387813(CHEMBL2058374)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387815(CHEMBL2058376)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387814(CHEMBL2058375)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387814(CHEMBL2058375)
Affinity DataIC50: 10.5nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387815(CHEMBL2058376)
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387816(CHEMBL2058377)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387816(CHEMBL2058377)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50117909(N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimet...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at type 1 angiotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387809(CHEMBL2058369)
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387809(CHEMBL2058369)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50117909(N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-ethyl-5,7-dimet...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at endothelin receptor subtype AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387808(CHEMBL2058368)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387808(CHEMBL2058368)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387807(CHEMBL2058367)
Affinity DataIC50: 45nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387807(CHEMBL2058367)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387806(CHEMBL2058366)
Affinity DataIC50: 92nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Bovine)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387806(CHEMBL2058366)
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50117910(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity at endothelin receptor subtype AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50117910(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataKi:  10nMAssay Description:Binding affinity at type 1 angiotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed