Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50040513
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human DYRK1A kinase expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333423(7-(Pyridin-3-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395379(CHEMBL2164712 | US9168247, CV12)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333416(7-(2-Methoxyethoxy)-1-methyl-beta-carboline | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395380(CHEMBL2164709 | US9168247, JR84)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395378(CHEMBL2164696 | US9168247, CV24)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed