Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50040520
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at KCNQ2/Q3 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395501(CHEMBL2163658)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395505(CHEMBL2164068)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM84184(SMR000688922 | cid_24248347 | MLS001143087 | 2-phe...)
Affinity DataIC50: 163nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395486(CHEMBL2163660)
Affinity DataEC50:  170nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395508(CHEMBL2164062)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 4(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at KCNQ4 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395481(CHEMBL2163667)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395500(CHEMBL2163659)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395518(CHEMBL2164049)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395498(CHEMBL2163662)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395515(CHEMBL2164054)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395506(CHEMBL2164066)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395514(CHEMBL2164055)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395488(CHEMBL1572950)
Affinity DataEC50:  350nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395507(CHEMBL2164064)
Affinity DataIC50: 360nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395499(CHEMBL2163661)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395502(CHEMBL2163657)
Affinity DataIC50: 390nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395497(CHEMBL2163664)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395504(CHEMBL2164069)
Affinity DataIC50: 470nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395493(CHEMBL2164065)
Affinity DataEC50:  490nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395491(CHEMBL1415708)
Affinity DataEC50:  700nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395496(CHEMBL1448089)
Affinity DataEC50:  743nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395484(CHEMBL2163663)
Affinity DataEC50:  800nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395489(CHEMBL2163656)
Affinity DataEC50:  950nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395495(CHEMBL2164050)
Affinity DataEC50:  990nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395473(CHEMBL2163666)
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395490(CHEMBL1732755)
Affinity DataEC50:  1.07E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM84166(N-2-biphenylyl-2-phenylbutanamide | MLS000575947 |...)
Affinity DataIC50: 1.32E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395492(CHEMBL2164067)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395494(CHEMBL2164063)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395485(CHEMBL1729184)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395516(CHEMBL2164053)
Affinity DataIC50: 2.22E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395487(CHEMBL1320944)
Affinity DataEC50:  2.35E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 2.92E+3nMAssay Description:Antagonist activity at KCNQ1 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395503(CHEMBL2163655)
Affinity DataIC50: 3.31E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395517(CHEMBL2164052)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395475(CHEMBL2163350)
Affinity DataIC50: 5.27E+3nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395471(CHEMBL2163670)
Affinity DataEC50:  7.09E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 8.12E+3nMAssay Description:Antagonist activity at KCNQ1/E1 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395472(CHEMBL2163668)
Affinity DataEC50:  8.66E+3nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395483(CHEMBL2163681)
Affinity DataEC50:  1.23E+4nMAssay Description:Agonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395479(CHEMBL2163673)
Affinity DataIC50: 1.27E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395474(CHEMBL2163686)
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50395509(CHEMBL2164061)
Affinity DataIC50: 2.02E+4nMAssay Description:Antagonist activity at KCNQ2 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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