Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50039876
TargetSerine/threonine-protein kinase Chk1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216171(pyrrolo[3',4':5,6]indolizino[8,7-b]indole-1,3-(2H,...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385583(CHEMBL2041917)
Affinity DataIC50: 90nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385585(CHEMBL2041919)
Affinity DataIC50: 130nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385583(CHEMBL2041917)
Affinity DataIC50: 180nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216159(5-hydroxy-pyrrolo[3',4':5,6]indolizino[8,7-b]indol...)
Affinity DataIC50: 200nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216159(5-hydroxy-pyrrolo[3',4':5,6]indolizino[8,7-b]indol...)
Affinity DataIC50: 260nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385580(CHEMBL2041914)
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385585(CHEMBL2041919)
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385584(CHEMBL2041918)
Affinity DataIC50: 420nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385583(CHEMBL2041917)
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216171(pyrrolo[3',4':5,6]indolizino[8,7-b]indole-1,3-(2H,...)
Affinity DataIC50: 520nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385584(CHEMBL2041918)
Affinity DataIC50: 910nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216171(pyrrolo[3',4':5,6]indolizino[8,7-b]indole-1,3-(2H,...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385585(CHEMBL2041919)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385579(CHEMBL2041749)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385584(CHEMBL2041918)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216171(pyrrolo[3',4':5,6]indolizino[8,7-b]indole-1,3-(2H,...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385580(CHEMBL2041914)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50216159(5-hydroxy-pyrrolo[3',4':5,6]indolizino[8,7-b]indol...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385581(CHEMBL2041915)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385580(CHEMBL2041914)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385579(CHEMBL2041749)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385579(CHEMBL2041749)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385578(CHEMBL2041912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385582(CHEMBL2041916)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385581(CHEMBL2041915)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385578(CHEMBL2041912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused rat recombinant DYRK1A expressed in Escherichia coli using Woodtide as substrate and [gamma-33P] after 30 mins by scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385582(CHEMBL2041916)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385578(CHEMBL2041912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385582(CHEMBL2041916)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using RS peptide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Paul Sabatier University

Curated by ChEMBL
LigandPNGBDBM50385581(CHEMBL2041915)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed