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Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50040028
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388123(CHEMBL2058762)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388127(CHEMBL2058758)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388125(CHEMBL2058756)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388115(CHEMBL2058975)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388126(CHEMBL2058757)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388115(CHEMBL2058975)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388118(CHEMBL2058970)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388122(CHEMBL2058761)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388113(CHEMBL2058973)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388119(CHEMBL2058972)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388123(CHEMBL2058762)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388119(CHEMBL2058972)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388127(CHEMBL2058758)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388125(CHEMBL2058756)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388114(CHEMBL2058974)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388126(CHEMBL2058757)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388114(CHEMBL2058974)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388121(CHEMBL2058760)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388113(CHEMBL2058973)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50: 0.920nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388117(CHEMBL2058969)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388117(CHEMBL2058969)
Affinity DataIC50: 1nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388122(CHEMBL2058761)
Affinity DataIC50: 1.03nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388121(CHEMBL2058760)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388124(CHEMBL2058967)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388120(CHEMBL2058759)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388118(CHEMBL2058970)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388124(CHEMBL2058967)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388120(CHEMBL2058759)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206038(((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388116(CHEMBL2058968)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388116(CHEMBL2058968)
Affinity DataIC50: 3nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206038(((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50: 12.2nMAssay Description:Inhibition of human recombinant DPP8 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206038(((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrol...)
Affinity DataIC50: 30.2nMAssay Description:Inhibition of human recombinant DPP9 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50: 72.4nMAssay Description:Inhibition of human recombinant DPP8 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50: 105nMAssay Description:Inhibition of human recombinant DPP9 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed