Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50040121
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50389436(CHEMBL1501622)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli using Z-MAL as substrate after 6 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM17471(3-(1H-1,2,3-triazol-5-yl)pyridine | 1,2,3-triazole...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli using Z-MAL as substrate after 6 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM27507(pyridine-3-carboxamide | nicotinamide | 3-Pyridine...)
Affinity DataIC50: 3.77E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli using Z-MAL as substrate after 6 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed