Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50040232
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataIC50: 9.91E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataIC50: 9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataIC50: 1.61E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataIC50: 1.96E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataIC50: 2.05E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataIC50: 3.24E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  7.04E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  7.07E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataKi:  7.19E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataKi:  7.51E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataKi:  7.74E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-7(Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataKi:  8.03E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataKi:  2.00E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataKi:  3.57E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed