Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50040633
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50005944(2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)
Affinity DataIC50: 200nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397451(CHEMBL2170736)
Affinity DataIC50: 300nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397448(CHEMBL2170728)
Affinity DataIC50: 800nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397452(CHEMBL520938)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397450(CHEMBL2170821)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50397449(CHEMBL2170832)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed