Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50040788
TargetCarbonic anhydrase 2(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 29nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase-2 assessed as hydrolysis of 4-nitrophenylacetateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400206(CHEMBL2180993)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50206554(N-(4-fluoro-benzyl)-N'-hydroxy-2-[1-phenyl-meth-(Z...)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400205(CHEMBL2180998)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400204(CHEMBL2180992)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400203(CHEMBL2180991)
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400202(CHEMBL2180995)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50206556(N1-(4-fluorobenzyl)-2-benzyl-N3-hydroxymalonamide ...)
Affinity DataIC50: 3.62E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400201(CHEMBL2180994)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400200(CHEMBL2180996)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400199(CHEMBL2180997)
Affinity DataIC50: 4.55E+3nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50400198(CHEMBL572368)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50062474(N1,2-dibenzyl-N3-hydroxymalonamide | 2,N-Dibenzyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50206555(2-[1-Phenyl-meth-(Z)-ylidene]-malonic Acid Monoeth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine kidney microsomal neutral aminopeptidase using Leu-pNA as substrate preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed