Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50042321
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Human)
University of Bayreuth
Curated by ChEMBL
University of Bayreuth
Curated by ChEMBL
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human Sirt5 deacetylation activity using FKRGVL-acetylLys-EYGVKV as substrate after 60 mins by glutamate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Human)
University of Bayreuth
Curated by ChEMBL
University of Bayreuth
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of human Sirt5 desuccinylation activity using SKEYFS-succinylLys-QK as substrate measured for 15 mins by MS analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Human)
University of Bayreuth
Curated by ChEMBL
University of Bayreuth
Curated by ChEMBL
Affinity DataIC50: 9.78E+4nMAssay Description:Inhibition of human Sirt5 deacetylation activity using FKRGVL-acetylLys-EYGVKV as substrate measured for 15 mins by MS analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Human)
University of Bayreuth
Curated by ChEMBL
University of Bayreuth
Curated by ChEMBL
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human Sirt5 deacetylation activity using SKEYFS-acetylLys-QK as substrate measured for 15 mins by MS analysisMore data for this Ligand-Target Pair
