Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50042482
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426654(CHEMBL2326202)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426655(CHEMBL2326201)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426656(CHEMBL2326200)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426657(CHEMBL2326199)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426653(CHEMBL2326203)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426654(CHEMBL2326202)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426655(CHEMBL2326201)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426656(CHEMBL2326200)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426657(CHEMBL2326199)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426653(CHEMBL2326203)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells coexpressing Galpha protein 16z25 assessed as increase in calcium mobilization measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426656(CHEMBL2326200)
Affinity DataKi:  0.0730nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426657(CHEMBL2326199)
Affinity DataKi:  0.291nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.296nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426653(CHEMBL2326203)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.429nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426655(CHEMBL2326201)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426654(CHEMBL2326202)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]melatonin from human MT2 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426655(CHEMBL2326201)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426653(CHEMBL2326203)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426656(CHEMBL2326200)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426654(CHEMBL2326202)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Hong Kong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50426657(CHEMBL2326199)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]melatonin from human MT1 receptor expressed in CHO cells after 60 mins by microbeta scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed