Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50042388
TargetGastrin-releasing peptide receptor(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50015490(NPY, human, rat | CHEMBL438945 | NPY | H-YPSKPDNPG...)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425232(CHEMBL2314836)
Affinity DataIC50: 9.80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50: 74nMAssay Description:Binding affinity to Y1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50: 80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed