Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50042652
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Staphylococcus aureus RN6390B Agr-mediated RNA3 promoter activation measured up to 6 hrs by Northern blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM11979(MgrA inhibitor, 1 | CHEMBL115145 | 5-[(3-carboxy-4...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Staphylococcus aureus Newman His6-tagged MgrA expressed in Escherichia coli BL21(DE3) using 5'-6-F-TAAACAACAAGTTGTCCAAA-3' as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM81554(MgrA inhibitor, 3)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Staphylococcus aureus Newman His6-tagged MgrA expressed in Escherichia coli BL21(DE3) using 5'-6-F-TAAACAACAAGTTGTCCAAA-3' as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM81553(MgrA inhibitor, 2)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Staphylococcus aureus Newman His6-tagged MgrA expressed in Escherichia coli BL21(DE3) using 5'-6-F-TAAACAACAAGTTGTCCAAA-3' as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM81555(MgrA inhibitor, 4)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Staphylococcus aureus Newman His6-tagged MgrA expressed in Escherichia coli BL21(DE3) using 5'-6-F-TAAACAACAAGTTGTCCAAA-3' as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed