Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50042668
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429068(CHEMBL2335740)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataEC50:  5nMAssay Description:Agonist activity at dopamine D1 receptor (unknown origin) transfected in CHO cell membranes assessed as increase in cAMP level after 8 mins by flash ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) transfected in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429068(CHEMBL2335740)
Affinity DataEC50:  8nMAssay Description:Agonist activity at dopamine D1 receptor (unknown origin) transfected in CHO cell membranes assessed as increase in cAMP level after 8 mins by flash ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataEC50:  11nMAssay Description:Agonist activity at dopamine D1 receptor (unknown origin) transfected in CHO cell membranes assessed as increase in cAMP level after 8 mins by flash ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429068(CHEMBL2335740)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429066(CHEMBL2335741)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) transfected in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429064(CHEMBL2335738)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429067(CHEMBL2335737)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) transfected in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429066(CHEMBL2335741)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429064(CHEMBL2335738)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429066(CHEMBL2335741)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) transfected in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429065(CHEMBL2331599)
Affinity DataEC50:  750nMAssay Description:Agonist activity at dopamine D1 receptor (unknown origin) transfected in CHO cell membranes assessed as increase in cAMP level after 8 mins by flash ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429069(CHEMBL2335736)
Affinity DataIC50: 840nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429064(CHEMBL2335738)
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) transfected in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429063(CHEMBL2335739)
Affinity DataKi:  3.34E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50429063(CHEMBL2335739)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin) expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed