Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50042686
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429392(CHEMBL2336766)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429400(CHEMBL2336769)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429399(CHEMBL2336753)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429398(CHEMBL2336759)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429397(CHEMBL2336760)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429396(CHEMBL2336761)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429395(CHEMBL2336762)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429394(CHEMBL2336764)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429393(CHEMBL2336765)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429383(CHEMBL2336758)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429391(CHEMBL2336767)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429390(CHEMBL2336768)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429389(CHEMBL2336770)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429388(CHEMBL2336771)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429387(CHEMBL2336754)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429386(CHEMBL2336755)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429385(CHEMBL2336756)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50429384(CHEMBL2336757)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed